Direct evidence for GPCR heterodimerization came from studies with non-functional GABA B receptors that dimerize to generate a functional receptor. Recent studies have also provided direct ...

Brohan, Janette and Goudra, Basavana G. 2017. The Role of GABA Receptor Agonists in Anesthesia and Sedation. CNS Drugs, Vol. 31, Issue. 10, p. 845. This concise, evidence-based board review book, ...

to specifically target the α5 subunit of GABA-A receptors in Ts65Dn mice, a classical animal model of DS. They found that the drug had no convulsant effects and did not promote any side effects ...

These sleeping pills work on the GABA receptors in the brain, which help control our level of alertness or relaxation. The selective GABA medications target only a certain type of GABA receptor ...

However, the development of antireflux compounds during the past 5 years (mainly GABA B agonists and mGluR5-negative ... Metabotropic glutamate receptor 5; MPEP: 2-methyl-6-(phenylethynyl ...