Diprenorphine - Wikipedia
Diprenorphine is a weak opioid antagonist used in veterinary medicine to reverse the effects of super-potent opioids like etorphine and carfentanil. It is also a partial agonist of the opioid receptors and can produce sedation and hallucinations in humans.
Diprenorphine: Uses, Interactions, Mechanism of Action
2007年7月31日 · Diprenorphine may increase the opioid antagonism activities of Naloxegol. Naltrexone The therapeutic efficacy of Naltrexone can be decreased when used in combination with Diprenorphine.
Use of butorphanol and diprenorphine to counter respiratory …
Today, butorphanol and diprenorphine are the most widely accessible of the opioid agonist-antagonists, but conflicting opinions exist as to which drug, or combination of drugs, provides the best respiratory support for immobilised white rhinoceroses.
Diprenorphine - an overview | ScienceDirect Topics
Diprenorphine is a weak opiate receptor partial agonist with similar in vivo affinities for the mu, kappa, and delta receptor subtypes.
Diprenorphine | C26H35NO4 | CID 443408 - PubChem
Diprenorphine is indicated to reverse the effects of powerful opioids including etorphine and carfentanil, often used for tranquilizing large animals. This drug is not approved for use in humans.
Diprenorphine - an overview | ScienceDirect Topics
Diprenorphine is a weak opiate receptor partial agonist that binds to the mu, kappa, and delta receptor subtypes, and it is used to study the role of opioid receptors in certain neurological conditions.
Diprenorphine - Wikiwand
Diprenorphine (brand name Revivon; former developmental code name M5050), also known as diprenorfin, is a non-selective, high- affinity, weak partial agonist of the μ- (MOR), κ- (KOR), and δ-opioid receptor (DOR) (with equal affinity) which …
DIPRENORPHINE - National Center for Advancing Translational …
As a narcotic antagonist similar in action to naloxone, DIPRENORPHINE is used to remobilize animals after analgesia by super-potent opioid analgesics such as etorphine and carfentanil. It is not used in humans.
Diprenorphine - an overview | ScienceDirect Topics
Diprenorphine is a nonspecific opioid antagonist that can be labeled with 11 C or 18 F for PET imaging of opioid receptors. It is also used to study opioid dysfunction in movement disorders such as Parkinson's disease and striatal neurodegeneration.
[6-O-methyl-11C]Diprenorphine - DrugBank Online
Diprenorphine is a highly potent and nonselective opioid receptors antagonist with subnanomolar affinity (7). Diprenorphine has been labeled as [6-O-methyl-11C]diprenorphine ([11C]DPN) (15, 16). [11C]DPN is being developed as a PET agent for …